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Angiogenic Host Defense Peptide AG-30/5C and Bradykinin B(2) receptor antagonist Icatibant are G protein-biased agonists for MRGPRX2 in mast cells

AG-30/5C is an angiogenic host defense peptide (HDP) that activates human mast cells (MC) via an unknown mechanism. Using shRNA-silenced human MC line (LAD2) and stably transfected RBL-2H3 cells, we demonstrate that AG-30/5C induces MC degranulation via Mas-related G protein coupled receptor (GPCR)...

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Detaylı Bibliyografya
Yayımlandı:J Immunol
Asıl Yazarlar: Roy, Saptarshi, Ganguly, Anirban, Haque, Maureen, Ali, Hydar
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: 2019
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6369923/
https://ncbi.nlm.nih.gov/pubmed/30651343
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.4049/jimmunol.1801227
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