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Design and Evaluation of Heterobivalent PAR1–PAR2 Ligands as Antagonists of Calcium Mobilization

[Image: see text] A novel class of bivalent ligands targeting putative protease-activated receptor (PAR) heteromers has been prepared based upon reported antagonists for the subtypes PAR1 and PAR2. Modified versions of the PAR1 antagonist RWJ-58259 containing alkyne adapters were connected via cyclo...

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Bibliografski detalji
Izdano u:ACS Med Chem Lett
Glavni autori: Majewski, Mark W., Gandhi, Disha M., Rosas, Ricardo, Kodali, Revathi, Arnold, Leggy A., Dockendorff, Chris
Format: Artigo
Jezik:Inglês
Izdano: American Chemical Society 2018
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC6331166/
https://ncbi.nlm.nih.gov/pubmed/30655958
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00538
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