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Organoruthenium(II) complexes of acetazolamide potently inhibit human carbonic anhydrase isoforms I, II, IX and XII

Two acetazolamide (AAZ) complexes with ruthenium(II) η(6)-p-cymene chloride were synthesised, characterised and tested for their inhibitory effects on several carbonic anhydrase (CA, EC 4.2.1.1) isoforms with pharmacological applications. Against human (h) isoform hCA I, the two complexes showed inh...

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Bibliografske podrobnosti
izdano v:J Enzyme Inhib Med Chem
Main Authors: Seršen, Sara, Traven, Katja, Kljun, Jakob, Turel, Iztok, Supuran, Claudiu T.
Format: Artigo
Jezik:Inglês
Izdano: Taylor & Francis 2019
Teme:
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC6327979/
https://ncbi.nlm.nih.gov/pubmed/30734595
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2018.1547288
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