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6’-Fluoro[4.3.0]bicyclo nucleic acid: synthesis, biophysical properties and molecular dynamics simulations

Here we report on the synthesis, biophysical properties and molecular modeling of oligonucleotides containing unsaturated 6’-fluoro[4.3.0]bicyclo nucleotides (6’F-bc(4,3)-DNA). Two 6’F-bc(4,3) phosphoramidite building blocks (T and C) were synthesized starting from a previously described [3.3.0]bicy...

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Pubblicato in:Beilstein J Org Chem
Autori principali: Frei, Sibylle, Istrate, Andrei, Leumann, Christian J
Natura: Artigo
Lingua:Inglês
Pubblicazione: Beilstein-Institut 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6317435/
https://ncbi.nlm.nih.gov/pubmed/30643586
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.14.288
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