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Improving Prediction Accuracy of Binding Free Energies and Poses of HIV Integrase Complexes Using the Binding Energy Distribution Analysis Method with Flattening Potentials

To accelerate conformation sampling of slow dynamics from receptor or ligand, we introduced flattening potentials on selected bonded and nonbonded intramolec-ular interactions to the binding energy distribution analysis method (BEDAM) for calculating absolute binding free energies of protein-ligand...

Deskribapen osoa

Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:J Chem Inf Model
Egile Nagusiak: Xia, Junchao, Flynn, William, Levy, Ronald M.
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: 2018
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6287956/
https://ncbi.nlm.nih.gov/pubmed/29927237
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.jcim.8b00194
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