Laddar...

Synthesis of Chiral, Enantiopure Allylic Amines by the Julia Olefination of α-Amino Esters

The four-step conversion of a series of N-Boc-protected l-amino acid methyl esters into enantiopure N-Boc allylamines by a modified Julia olefination is described. Key steps include the reaction of a lithiated phenylalkylsulfone with amino esters, giving chiral β-ketosulfones, and the reductive elim...

Full beskrivning

Sparad:
Bibliografiska uppgifter
I publikationen:Molecules
Huvudupphovsmän: Benedetti, Fabio, Berti, Federico, Fanfoni, Lidia, Garbo, Michele, Regini, Giorgia, Felluga, Fulvia
Materialtyp: Artigo
Språk:Inglês
Publicerad: MDPI 2016
Ämnen:
Länkar:https://ncbi.nlm.nih.gov/pmc/articles/PMC6273449/
https://ncbi.nlm.nih.gov/pubmed/27338326
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules21060805
Taggar: Lägg till en tagg
Inga taggar, Lägg till första taggen!