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Practical and Efficient Synthesis of α-Aminophosphonic Acids Containing 1,2,3,4-Tetrahydroquinoline or 1,2,3,4-Tetrahydroisoquinoline Heterocycles

We report here a practical and efficient synthesis of α-aminophosphonic acid incorporated into 1,2,3,4-tetrahydroquinoline and 1,2,3,4-tetrahydroisoquinoline heterocycles, which could be considered to be conformationally constrained analogues of pipecolic acid. The principal contribution of this syn...

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Publicat a:Molecules
Autors principals: Ordóñez, Mario, Arizpe, Alicia, Sayago, Fracisco J., Jiménez, Ana I., Cativiela, Carlos
Format: Artigo
Idioma:Inglês
Publicat: MDPI 2016
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6273407/
https://ncbi.nlm.nih.gov/pubmed/27589713
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/molecules21091140
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