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(Radio)Fluoro-Click Reaction Enabled by a Hydrogen Bonding Cluster

We have developed a widely applicable nucleophilic (radio)fluoro-click reaction of ynamides with readily available and easy handling KF((18)F). The reactions exhibited high functional group tolerance and needed only ambient atmosphere. Most importantly, this is the first (18)F addition protocol to C...

Disgrifiad llawn

Wedi'i Gadw mewn:
Manylion Llyfryddiaeth
Cyhoeddwyd yn:Angew Chem Int Ed Engl
Prif Awduron: Zeng, Xiaojun, Li, Junling, Ng, Chin K., Hammond, Gerald B., Xu, Bo
Fformat: Artigo
Iaith:Inglês
Cyhoeddwyd: 2018
Pynciau:
Mynediad Ar-lein:https://ncbi.nlm.nih.gov/pmc/articles/PMC6233894/
https://ncbi.nlm.nih.gov/pubmed/29276938
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/anie.201711341
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