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Carbonic anhydrase inhibition with a series of novel benzenesulfonamide-triazole conjugates

We report the synthesis and characterisation of a novel series of triazole benzenesulfonamide derivatives, which incorporate the general pharmacophore associated with carbonic anhydrase (CA, EC 4.2.1.1) inhibitors. The synthesised compounds were tested in vitro against four human carbonic anhydrase...

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Detaylı Bibliyografya
Yayımlandı:J Enzyme Inhib Med Chem
Asıl Yazarlar: El-Gazzar, Marwa G., Nafie, Nessma H., Nocentini, Alessio, Ghorab, Mostafa M., Heiba, Helmi I., Supuran, Claudiu T.
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Taylor & Francis 2018
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6171417/
https://ncbi.nlm.nih.gov/pubmed/30274535
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1080/14756366.2018.1513927
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