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Preparation of a Crystalline Salt of Indomethacin and Tromethamine by Hot Melt Extrusion Technology

Although salt formation is the most ubiquitous and effective method of increasing the solubility and dissolution rates of acidic and basic drugs, it consumes large quantities of organic solvents and is a batch process. Herein, we show that the dissolution rate of indomethacin (a poorly water-soluble...

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Dades bibliogràfiques
Publicat a:Eur J Pharm Biopharm
Autors principals: Bookwala, Mustafa, Thipsay, Priyanka, Ross, Samir, Zhang, Feng, Bandari, Suresh, Repka, Michael A.
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6154477/
https://ncbi.nlm.nih.gov/pubmed/30086393
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.ejpb.2018.08.001
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