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PF-06827443 Displays Robust Allosteric Agonist and Positive Allosteric Modulator Activity in High Receptor Reserve and Native Systems

Positive allosteric modulators (PAMs) of the M(1) subtype of muscarinic acetylcholine receptor have attracted intense interest as an exciting new approach for improving the cognitive deficits in schizophrenia and Alzheimer’s disease. Recent evidence suggests that the presence of intrinsic agonist ac...

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Библиографические подробности
Опубликовано в: :ACS Chem Neurosci
Главные авторы: Moran, Sean P., Cho, Hyekyung P., Maksymetz, James, Remke, Daniel H., Hanson, Ryan M., Niswender, Colleen M., Lindsley, Craig W., Rook, Jerri M., Conn, P. Jeffrey
Формат: Artigo
Язык:Inglês
Опубликовано: 2018
Предметы:
Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC6146053/
https://ncbi.nlm.nih.gov/pubmed/29683646
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.8b00106
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