載入...

Peptidomimetics for Targeting Protein–Protein Interactions between DOT1L and MLL Oncofusion Proteins AF9 and ENL

[Image: see text] MLL-fusion proteins, AF9 and ENL, play an essential role in the recruitment of DOT1L and the H3K79 hypermethylation of MLL target genes, which is pivotal for leukemogenesis. Blocking these interactions may represent a novel therapeutic approach for MLL-rearranged leukemia. Based on...

全面介紹

Na minha lista:
書目詳細資料
發表在:ACS Med Chem Lett
Main Authors: Du, Lei, Grigsby, Sierrah M., Yao, Aihong, Chang, Yujie, Johnson, Garrett, Sun, Haiying, Nikolovska-Coleska, Zaneta
格式: Artigo
語言:Inglês
出版: American Chemical Society 2018
在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC6142068/
https://ncbi.nlm.nih.gov/pubmed/30258537
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00175
標簽: 添加標簽
沒有標簽, 成為第一個標記此記錄!