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NOP receptor pharmacological profile – A dynamic mass redistribution study

The Nociceptin/Orphanin FQ (N/OFQ) peptide NOP receptor is coupled to pertussis toxin (PTX)-sensitive G proteins (G(i/o)) whose activation leads to the inhibition of both cAMP production and calcium channel activity, and to the stimulation of potassium currents. The label free dynamic mass redistrib...

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Dettagli Bibliografici
Pubblicato in:PLoS One
Autori principali: Malfacini, Davide, Simon, Katharina, Trapella, Claudio, Guerrini, Remo, Zaveri, Nurulain T., Kostenis, Evi, Calo’, Girolamo
Natura: Artigo
Lingua:Inglês
Pubblicazione: Public Library of Science 2018
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6117024/
https://ncbi.nlm.nih.gov/pubmed/30161182
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1371/journal.pone.0203021
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