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Binding kinetics of cariprazine and aripiprazole at the dopamine D(3) receptor

The dissociation behaviours of aripiprazole and cariprazine at the human D(2) and D(3) receptor are evaluated. A potential correlation between kinetics and in vivo profiles, especially cariprazine’s action on negative symptoms in schizophrenia, is investigated. The binding kinetics of four ligands w...

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Publicat a:Sci Rep
Autors principals: Frank, Annika, Kiss, Dóra J., Keserű, György M., Stark, Holger
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2018
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC6104066/
https://ncbi.nlm.nih.gov/pubmed/30131592
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-30794-y
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