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Disruption of Amino Acid Homeostasis by Novel ASCT2 Inhibitors Involves Multiple Targets

The glutamine transporter ASCT2 (SLC1A5) is actively investigated as an oncological target, but the field lacks efficient ASCT2 inhibitors. A new group of ASCT2 inhibitors, 2-amino-4-bis(aryloxybenzyl)aminobutanoic acids (AABA), were developed recently and shown to suppress tumor growth in preclinic...

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Detaylı Bibliyografya
Yayımlandı:Front Pharmacol
Asıl Yazarlar: Bröer, Angelika, Fairweather, Stephen, Bröer, Stefan
Materyal Türü: Artigo
Dil:Inglês
Baskı/Yayın Bilgisi: Frontiers Media S.A. 2018
Konular:
Online Erişim:https://ncbi.nlm.nih.gov/pmc/articles/PMC6060247/
https://ncbi.nlm.nih.gov/pubmed/30072900
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3389/fphar.2018.00785
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