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Novel Aminoquinoline Derivatives Significantly Reduce Parasite Load in Leishmania infantum Infected Mice

[Image: see text] In this Letter, a detailed analysis of 30 4-aminoquinoline-based compounds with regard to their potential as antileishmanial drugs has been carried out. Ten compounds demonstrated IC(50) < 1 μM against promastigote stages of L. infantum and L. tropica, and five compounds showed...

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Detalhes bibliográficos
Publicado no:ACS Med Chem Lett
Main Authors: Konstantinović, Jelena, Videnović, Milica, Orsini, Stefania, Bogojević, Katarina, D’Alessandro, Sarah, Scaccabarozzi, Diletta, Terzić Jovanović, Nataša, Gradoni, Luigi, Basilico, Nicoletta, Šolaja, Bogdan A.
Formato: Artigo
Idioma:Inglês
Publicado em: American Chemical Society 2018
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC6047044/
https://ncbi.nlm.nih.gov/pubmed/30034591
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00053
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