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Chemical Strategies for Half-Life Extension of Biopharmaceuticals: Lipidation and Its Alternatives

[Image: see text] Strategies for half-life extension are often required in the design of new biopharmaceuticals. This Viewpoint focuses on chemical moieties that convey protraction by albumin binding or by self-assembly to form larger structures, with GLP-1 and insulin as examples.

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Bibliographic Details
Published in:ACS Med Chem Lett
Main Authors: Bech, Esben M., Pedersen, Søren L., Jensen, Knud J.
Format: Artigo
Language:Inglês
Published: American Chemical Society 2018
Online Access:https://ncbi.nlm.nih.gov/pmc/articles/PMC6047018/
https://ncbi.nlm.nih.gov/pubmed/30034579
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00226
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