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Aptamers as Therapeutics

Aptamers are single-stranded nucleic acid molecules that bind to and inhibit proteins and are commonly produced by systematic evolution of ligands by exponential enrichment (SELEX). Aptamers undergo extensive pharmacological revision, which alters affinity, specificity, and therapeutic half-life, ta...

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Pubblicato in:Annu Rev Pharmacol Toxicol
Autori principali: Nimjee, Shahid M., White, Rebekah R., Becker, Richard C., Sullenger, Bruce A.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC6035745/
https://ncbi.nlm.nih.gov/pubmed/28061688
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1146/annurev-pharmtox-010716-104558
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