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Aptamers as Therapeutics

Aptamers are single-stranded nucleic acid molecules that bind to and inhibit proteins and are commonly produced by systematic evolution of ligands by exponential enrichment (SELEX). Aptamers undergo extensive pharmacological revision, which alters affinity, specificity, and therapeutic half-life, ta...

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Detalles Bibliográficos
Publicado en:Annu Rev Pharmacol Toxicol
Autores principales: Nimjee, Shahid M., White, Rebekah R., Becker, Richard C., Sullenger, Bruce A.
Formato: Artigo
Lenguaje:Inglês
Publicado: 2017
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Acceso en línea:https://ncbi.nlm.nih.gov/pmc/articles/PMC6035745/
https://ncbi.nlm.nih.gov/pubmed/28061688
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1146/annurev-pharmtox-010716-104558
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