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Effect of Methionine Oxidation and Substitution of α-Conotoxin TxID on α3β4 Nicotinic Acetylcholine Receptor

α-Conotoxin TxID was discovered from Conus textile by gene cloning, which has 4/6 inter-cysteine loop spacing and selectively inhibits α3β4 nicotinic acetylcholine receptor (nAChR) subtype. However, TxID is susceptible to modification due to it containing a methionine (Met) residue that easily forms...

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Gorde:
Xehetasun bibliografikoak
Argitaratua izan da:Mar Drugs
Egile Nagusiak: Ren, Jie, Li, Rui, Ning, Jiong, Zhu, Xiaopeng, Zhangsun, Dongting, Wu, Yong, Luo, Sulan
Formatua: Artigo
Hizkuntza:Inglês
Argitaratua: MDPI 2018
Gaiak:
Sarrera elektronikoa:https://ncbi.nlm.nih.gov/pmc/articles/PMC6025358/
https://ncbi.nlm.nih.gov/pubmed/29925760
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3390/md16060215
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