Loading...

Enantioselective phase-transfer catalyzed alkylation of 1-methyl-7-methoxy-2-tetralone: an effective route to dezocine

In order to prepare asymmetrically (R)-(+)-1-(5-bromopentyl)-1-methyl-7-methoxy-2-tetralone (3a), a key intermediate of dezocine, 17 cinchona alkaloid-derived catalysts were prepared and screened for the enantioselective alkylation of 1-methyl-7-methoxy-2-tetralone with 1,5-dibromopentane, and the b...

Fuld beskrivelse

Na minha lista:
Bibliografiske detaljer
Udgivet i:Beilstein J Org Chem
Main Authors: Li, Ruipeng, Liu, Zhenren, Chen, Liang, Pan, Jing, Zhou, Weicheng
Format: Artigo
Sprog:Inglês
Udgivet: Beilstein-Institut 2018
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC6009193/
https://ncbi.nlm.nih.gov/pubmed/29977405
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.3762/bjoc.14.119
Tags: Tilføj Tag
Ingen Tags, Vær først til at tagge denne postø!