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Design, synthesis and anti-tumor activity study of novel histone deacetylase inhibitors containing isatin-based caps and o-phenylenediamine-based zinc binding groups

As a hot topic of epigenetic studies, histone deacetylases (HDACs) are related to lots of diseases, especially cancer. Further researches indicated that different HDAC isoforms played various roles in a wide range of tumor types. Herein a novel series of HDAC inhibitors with isatin-based caps and o-...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Gao, Shuai, Zang, Jie, Gao, Qianwen, Liang, Xuewu, Ding, Qinge, Li, Xiaoyang, Xu, Wenfang, Chou, C. James, Zhang, Yingjie
Formato: Artigo
Idioma:Inglês
Publicado em: 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5994915/
https://ncbi.nlm.nih.gov/pubmed/28511906
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2017.03.036
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