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Design of small molecules that compete with nucleotide binding to an engineered oncogenic KRAS allele

RAS mutations are found in 30% of all human cancers, with KRAS the most frequently mutated among the three RAS isoforms (KRAS, NRAS, HRAS). However, directly targeting oncogenic KRAS with small molecules in the nucleotide-binding site has been difficult due to the high affinity of KRAS for GDP and G...

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Detalhes bibliográficos
Publicado no:Biochemistry
Main Authors: Zhang, Yan, Larraufie, Marie-Hélène, Musavi, Leila, Akkiraju, Hemanth, Brown, Lewis M., Stockwell, Brent
Formato: Artigo
Idioma:Inglês
Publicado em: 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5960803/
https://ncbi.nlm.nih.gov/pubmed/29313669
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.7b01113
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