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AICAR inhibits NFκB DNA binding independently of AMPK to attenuate LPS-triggered inflammatory responses in human macrophages

5-aminoimidazole-4-carboxamide-1-β-D-ribofuranoside (AICAR) is an established pharmacological activator of AMP-activated protein kinase (AMPK). Both, AICAR and AMPK were reported to attenuate inflammation. However, AICAR is known for many AMPK-independent effects, although the mechanisms remain inco...

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Опубликовано в: :Sci Rep
Главные авторы: Kirchner, Johannes, Brüne, Bernhard, Namgaladze, Dmitry
Формат: Artigo
Язык:Inglês
Опубликовано: Nature Publishing Group UK 2018
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Online-ссылка:https://ncbi.nlm.nih.gov/pmc/articles/PMC5958102/
https://ncbi.nlm.nih.gov/pubmed/29773845
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-018-26102-3
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