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Shaping Substrate Selectivity in a Broad-Spectrum Metallo-β-Lactamase

Metallo-β-lactamases (MBLs) are the major group of carbapenemases produced by bacterial pathogens. The design of MBL inhibitors has been limited by, among other issues, incomplete knowledge about how these enzymes modulate substrate recognition. While most MBLs are broad-spectrum enzymes, B2 MBLs ar...

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Dettagli Bibliografici
Pubblicato in:Antimicrob Agents Chemother
Autori principali: González, Lisandro J., Stival, Cintia, Puzzolo, Juan L., Moreno, Diego M., Vila, Alejandro J.
Natura: Artigo
Lingua:Inglês
Pubblicazione: American Society for Microbiology 2018
Soggetti:
Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5913924/
https://ncbi.nlm.nih.gov/pubmed/29358299
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.02079-17
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