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Targeting Ligandable Pockets on Plant Homeodomain (PHD) Zinc Finger Domains by a Fragment-Based Approach

[Image: see text] Plant homeodomain (PHD) zinc fingers are histone reader domains that are often associated with human diseases. Despite this, they constitute a poorly targeted class of readers, suggesting low ligandability. Here, we describe a successful fragment-based campaign targeting PHD finger...

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Bibliografske podrobnosti
izdano v:ACS Chem Biol
Main Authors: Amato, Anastasia, Lucas, Xavier, Bortoluzzi, Alessio, Wright, David, Ciulli, Alessio
Format: Artigo
Jezik:Inglês
Izdano: American Chemical Society 2018
Online dostop:https://ncbi.nlm.nih.gov/pmc/articles/PMC5913730/
https://ncbi.nlm.nih.gov/pubmed/29529862
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.7b01093
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