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A Review of Salvinorin Analogs and their Kappa-Opioid Receptor Activity

The plant metabolite salvinorin A potently and selectively agonizes the human kappa-opioid receptor, an emerging target for next-generation analgesics. Here we review analogs of the salvinorin chemotype and their effects on selectivity, affinity and potency. Extensive peripheral modifications using...

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書目詳細資料
發表在:Bioorg Med Chem Lett
Main Authors: Roach, Jeremy J., Shenvi, Ryan A.
格式: Artigo
語言:Inglês
出版: 2018
主題:
在線閱讀:https://ncbi.nlm.nih.gov/pmc/articles/PMC5912166/
https://ncbi.nlm.nih.gov/pubmed/29615341
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.03.029
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