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A Caged Enkephalin Optimized for Simultaneously Probing Mu and Delta Opioid Receptors

Physiological responses to the opioid neuropeptide enkephalin often involve both mu and delta opioid receptors. To facilitate quantitative studies into opioid signaling, we previously developed a caged [Leu(5)]-enkephalin that responds to ultraviolet irradiation, but its residual activity at delta r...

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Bibliografiske detaljer
Udgivet i:ACS Chem Neurosci
Main Authors: Banghart, Matthew R., He, Xinyi J., Sabatini, Bernardo L.
Format: Artigo
Sprog:Inglês
Udgivet: 2017
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5906201/
https://ncbi.nlm.nih.gov/pubmed/29266926
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.7b00485
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