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A Caged Enkephalin Optimized for Simultaneously Probing Mu and Delta Opioid Receptors

Physiological responses to the opioid neuropeptide enkephalin often involve both mu and delta opioid receptors. To facilitate quantitative studies into opioid signaling, we previously developed a caged [Leu(5)]-enkephalin that responds to ultraviolet irradiation, but its residual activity at delta r...

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Pubblicato in:ACS Chem Neurosci
Autori principali: Banghart, Matthew R., He, Xinyi J., Sabatini, Bernardo L.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5906201/
https://ncbi.nlm.nih.gov/pubmed/29266926
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.7b00485
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