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A Caged Enkephalin Optimized for Simultaneously Probing Mu and Delta Opioid Receptors

Physiological responses to the opioid neuropeptide enkephalin often involve both mu and delta opioid receptors. To facilitate quantitative studies into opioid signaling, we previously developed a caged [Leu(5)]-enkephalin that responds to ultraviolet irradiation, but its residual activity at delta r...

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Détails bibliographiques
Publié dans:ACS Chem Neurosci
Auteurs principaux: Banghart, Matthew R., He, Xinyi J., Sabatini, Bernardo L.
Format: Artigo
Langue:Inglês
Publié: 2017
Sujets:
Accès en ligne:https://ncbi.nlm.nih.gov/pmc/articles/PMC5906201/
https://ncbi.nlm.nih.gov/pubmed/29266926
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschemneuro.7b00485
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