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In Vitro and In Vivo Investigation of Potential for Complex CYP3A Interaction for PF‐00251802 (Dagrocorat), a Novel Dissociated Agonist of the Glucocorticoid Receptor

The dissociated agonists of the glucocorticoid receptor are a novel class of agents in clinical development for rheumatoid arthritis. PF‐04171327 (fosdagrocorat) is a phosphate ester prodrug of PF‐00251802 (dagrocorat), a selective high‐affinity partial agonist of the glucocorticoid receptor, which...

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Detalhes bibliográficos
Publicado no:Clin Pharmacol Drug Dev
Main Authors: Ripp, Sharon L., Mukherjee, Arnab, Eng, Heather, Stock, Thomas, Fleishaker, Dona, Checchio, Tina, Tammara, Brinda
Formato: Artigo
Idioma:Inglês
Publicado em: John Wiley and Sons Inc. 2017
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5900965/
https://ncbi.nlm.nih.gov/pubmed/29112329
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/cpdd.411
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