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Dissociated Agonist of Glucocorticoid Receptor or Prednisone for Active Rheumatoid Arthritis: Effects on P1NP and Osteocalcin Pharmacodynamics

Fosdagrocorat (PF‐04171327), a dissociated agonist of the glucocorticoid receptor, has potent anti‐inflammatory activity in patients with rheumatoid arthritis with reduced adverse effects on bone health. To identify fosdagrocorat doses with bone formation marker changes similar to prednisone 5 mg, w...

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Dettagli Bibliografici
Pubblicato in:CPT Pharmacometrics Syst Pharmacol
Autori principali: Shoji, S, Suzuki, A, Conrado, DJ, Peterson, MC, Hey‐Hadavi, J, McCabe, D, Rojo, R, Tammara, BK
Natura: Artigo
Lingua:Inglês
Pubblicazione: John Wiley and Sons Inc. 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5529777/
https://ncbi.nlm.nih.gov/pubmed/28556506
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/psp4.12201
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