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Cannabinoid receptor interacting protein suppress agonist–driven CB(1) receptor internalization and regulates receptor replenishment in an agonist–biased manner

Cannabinoid receptor interacting protein 1a (CRIP1a) is a CB(1) receptor (CB(1)R) distal C-terminus-associated protein that modulates CB(1)R signaling via G proteins, and CB(1)R down-regulation but not desensitization (Blume et al. [2015] Cell Signal., 27, 716–726; Smith et al. [2015] Mol. Pharmacol...

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Dades bibliogràfiques
Publicat a:J Neurochem
Autors principals: Blume, Lawrence C., Leone-Kabler, Sandra, Luessen, Deborah J., Marrs, Glen S., Lyons, Erica, Bass, Caroline E., Chen, Rong, Selley, Dana E., Howlett, Allyn C.
Format: Artigo
Idioma:Inglês
Publicat: 2016
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5894350/
https://ncbi.nlm.nih.gov/pubmed/27513693
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/jnc.13767
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