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VKORC1 and VKORC1L1 have distinctly different oral anticoagulant dose-response characteristics and binding sites

Vitamin K reduction is catalyzed by 2 enzymes in vitro: the vitamin K 2,3-epoxide reductase complex subunit 1 (VKORC1) and its isozyme VKORC1-like1 (VKORC1L1). In vivo, VKORC1 reduces vitamin K to sustain γ-carboxylation of vitamin K-dependent proteins, including coagulation factors. Inhibition of V...

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Publicat a:Blood Adv
Autors principals: Czogalla, Katrin J., Liphardt, Kerstin, Höning, Klara, Hornung, Veit, Biswas, Arijit, Watzka, Matthias, Oldenburg, Johannes
Format: Artigo
Idioma:Inglês
Publicat: American Society of Hematology 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5873226/
https://ncbi.nlm.nih.gov/pubmed/29581108
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1182/bloodadvances.2017006775
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