Carregant...

A small group of sulfated benzofurans induces steady-state submaximal inhibition of thrombin

Despite the development of promising direct oral anticoagulants, which are all orthosteric inhibitors, a sizable number of patients suffer from bleeding complications. We have hypothesized that allosterism based on the heparin-binding exosites presents a major opportunity to induce sub-maximal inhib...

Descripció completa

Guardat en:
Dades bibliogràfiques
Publicat a:Bioorg Med Chem Lett
Autors principals: Afosah, Daniel K., Verespy, Stephen, Al-Horani, Rami A., Boothello, Rio S., Karuturi, Rajesh, Desai, Umesh R.
Format: Artigo
Idioma:Inglês
Publicat: 2018
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5851871/
https://ncbi.nlm.nih.gov/pubmed/29459207
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmcl.2018.01.069
Etiquetes: Afegir etiqueta
Sense etiquetes, Sigues el primer a etiquetar aquest registre!