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Inhibition of transcription factor-DNA complexes and gene expression by a microgonotropen

Developing minor groove-binding drugs to selectively inhibit transcription factor (TF)/DNA interactions and accompanying gene expression is a current goal in drug development studies. Equipping minor groove-binding agents with positively charged, major groove-contacting side chains yields microgonot...

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Autors principals: White, Christine M., Satz, Alexander L., Bruice, Thomas C., Beerman, Terry A.
Format: Artigo
Idioma:Inglês
Publicat: The National Academy of Sciences 2001
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Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC58510/
https://ncbi.nlm.nih.gov/pubmed/11535831
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1073/pnas.191374698
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