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Mutation in the FGFR1 tyrosine kinase domain or inactivation of PTEN is associated with acquired resistance to FGFR inhibitors in FGFR1-driven leukemia/lymphomas

Stem cell leukemia/lymphoma syndrome (SCLL) is driven by constitutive activation of chimeric FGFR1 kinases generated by chromosome translocations. We have shown that FGFR inhibitors significantly suppress leukemia and lymphoma development in vivo, and cell viability in vitro. Since resistance to tar...

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Detalles Bibliográficos
Publicado en:Int J Cancer
Main Authors: Cowell, John K, Qin, Haiyan, Hu, Tianxiang, Wu, Qing, Bhole, Aaron, Ren, Mingqiang
Formato: Artigo
Idioma:Inglês
Publicado: 2017
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Acceso en liña:https://ncbi.nlm.nih.gov/pmc/articles/PMC5850950/
https://ncbi.nlm.nih.gov/pubmed/28646488
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1002/ijc.30848
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