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Stereochemical Structure Activity Relationship Studies (S-SAR) of Tetrahydrolipstatin

[Image: see text] Tetrahydrolipstatin (THL), its enantiomer, and an additional six diastereomers were evaluated as inhibitors of the hydrolysis of p-nitrophenyl butyrate by porcine pancreatic lipase. IC(50)s were found for all eight stereoisomers ranging from a low of 4.0 nM for THL to a high of 930...

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Vydáno v:ACS Med Chem Lett
Hlavní autoři: Liu, Xiaofan, Wang, Yanping, Duclos, Richard I., O’Doherty, George A.
Médium: Artigo
Jazyk:Inglês
Vydáno: American Chemical Society 2018
On-line přístup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5846039/
https://ncbi.nlm.nih.gov/pubmed/29541373
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acsmedchemlett.8b00050
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