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Metabolic Profiling of the Novel Hypoxia-Inducible Factor 2α Inhibitor PT2385 In Vivo and In Vitro

PT2385 is a first-in-class, selective small-molecule inhibitor of hypoxia-inducible factor-2α (HIF-2α) developed for the treatment of advanced clear cell renal cell carcinoma. Preclinical results demonstrated that PT2385 has potent antitumor efficacy in mouse xenograft models of kidney cancer. It al...

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Detalhes bibliográficos
Publicado no:Drug Metab Dispos
Main Authors: Xie, Cen, Gao, Xiaoxia, Sun, Dongxue, Zhang, Youbo, Krausz, Kristopher W., Qin, Xuemei, Gonzalez, Frank J.
Formato: Artigo
Idioma:Inglês
Publicado em: The American Society for Pharmacology and Experimental Therapeutics 2018
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5829541/
https://ncbi.nlm.nih.gov/pubmed/29363499
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1124/dmd.117.079723
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