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Parasite-Mediated Degradation of Synthetic Ozonide Antimalarials Impacts In Vitro Antimalarial Activity

The peroxide bond of the artemisinins inspired the development of a class of fully synthetic 1,2,4-trioxolane-based antimalarials, collectively known as the ozonides. Similar to the artemisinins, heme-mediated degradation of the ozonides generates highly reactive radical species that are thought to...

Ausführliche Beschreibung

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Bibliographische Detailangaben
Veröffentlicht in:Antimicrob Agents Chemother
Hauptverfasser: Giannangelo, Carlo, Stingelin, Lukas, Yang, Tuo, Tilley, Leann, Charman, Susan A., Creek, Darren J.
Format: Artigo
Sprache:Inglês
Veröffentlicht: American Society for Microbiology 2018
Schlagworte:
Online Zugang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5826100/
https://ncbi.nlm.nih.gov/pubmed/29263074
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1128/AAC.01566-17
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