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Mechanisms of Proton Relay and Product Release by Class A β-Lactamase at Ultrahigh Resolution

The β-lactam antibiotics inhibit penicillin-binding proteins (PBPs) by forming a stable, covalent, acyl-enzyme complex. During the evolution from PBPs to Class A β-lactamases, the β-lactamases acquired Glu166 to activate a catalytic water and cleave the acyl-enzyme bond. Here we present three produc...

Täydet tiedot

Tallennettuna:
Bibliografiset tiedot
Julkaisussa:FEBS J
Päätekijät: Lewandowski, Eric M., Lethbridge, Kathryn G., Sanishvili, Ruslan, Skiba, Joanna, Kowalski, Konrad, Chen, Yu
Aineistotyyppi: Artigo
Kieli:Inglês
Julkaistu: 2017
Aiheet:
Linkit:https://ncbi.nlm.nih.gov/pmc/articles/PMC5760336/
https://ncbi.nlm.nih.gov/pubmed/29095570
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1111/febs.14315
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