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How Oliceridine (TRV-130) Binds and Stabilizes a μ-Opioid Receptor Conformational State That Selectively Triggers G Protein Signaling Pathways

Substantial attention has recently been devoted to G protein-biased agonism of the μ-opioid receptor (MOR) as an ideal new mechanism for the design of analgesics devoid of serious side effects. However, designing opioids with appropriate efficacy and bias is challenging because it requires an unders...

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Detalhes bibliográficos
Publicado no:Biochemistry
Main Authors: Schneider, Sebastian, Provasi, Davide, Filizola, Marta
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5745009/
https://ncbi.nlm.nih.gov/pubmed/27778501
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acs.biochem.6b00948
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