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The Sam-Sam interaction between Ship2 and the EphA2 receptor: design and analysis of peptide inhibitors

The lipid phosphatase Ship2 represents a drug discovery target for the treatment of different diseases, including cancer. Its C-terminal sterile alpha motif domain (Ship2-Sam) associates with the Sam domain from the EphA2 receptor (EphA2-Sam). This interaction is expected to mainly induce pro-oncoge...

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Dades bibliogràfiques
Publicat a:Sci Rep
Autors principals: Mercurio, Flavia Anna, Di Natale, Concetta, Pirone, Luciano, Iannitti, Roberta, Marasco, Daniela, Pedone, Emilia Maria, Palumbo, Rosanna, Leone, Marilisa
Format: Artigo
Idioma:Inglês
Publicat: Nature Publishing Group UK 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5727260/
https://ncbi.nlm.nih.gov/pubmed/29234063
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-17684-5
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