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Global profiling of lysine reactivity and ligandability in the human proteome

Nucleophilic amino acids make important contributions to protein function, including performing key roles in catalysis and serving as sites for post-translational modification. Electrophilic groups that target amino-acid nucleophiles have been used to create covalent ligands and drugs, but have, so...

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Dettagli Bibliografici
Pubblicato in:Nat Chem
Autori principali: Hacker, Stephan M., Backus, Keriann M., Lazear, Michael R., Forli, Stefano, Correia, Bruno E., Cravatt, Benjamin F.
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5726523/
https://ncbi.nlm.nih.gov/pubmed/29168484
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchem.2826
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