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Structural Flexibility of an Inhibitor Overcomes Drug Resistance Mutations in Staphylococcus aureus FtsZ

In the effort to combat antibiotic resistance, inhibitors of the essential bacterial protein FtsZ have emerged as a promising new class of compounds with clinical potential. One such FtsZ inhibitor (TXA707) is associated with potent activity against clinical isolates of methicillin-resistant Staphyl...

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Dettagli Bibliografici
Pubblicato in:ACS Chem Biol
Autori principali: Fujita, Junso, Maeda, Yoko, Mizohata, Eiichi, Inoue, Tsuyoshi, Kaul, Malvika, Parhi, Ajit K., LaVoie, Edmond J., Pilch, Daniel S., Matsumura, Hiroyoshi
Natura: Artigo
Lingua:Inglês
Pubblicazione: 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5705026/
https://ncbi.nlm.nih.gov/pubmed/28621933
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1021/acschembio.7b00323
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