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Design and synthesis of triarylacrylonitrile analogues of tamoxifen with improved binding selectivity to protein kinase C

The clinical selective estrogen receptor modulator tamoxifen is also a modest inhibitor of protein kinase C, a target implicated in several untreatable brain diseases such as amphetamine abuse. This inhibition and tamoxifen’s ability to cross the blood brain barrier make it an attractive scaffold to...

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Detalhes bibliográficos
Publicado no:Bioorg Med Chem
Main Authors: Carpenter, Colleen, Sorenson, Roderick J., Jin, Yafei, Klossowski, Szymon, Cierpicki, Tomascz, Gnegy, Margaret, Showalter, Hollis D.
Formato: Artigo
Idioma:Inglês
Publicado em: 2016
Assuntos:
Acesso em linha:https://ncbi.nlm.nih.gov/pmc/articles/PMC5696786/
https://ncbi.nlm.nih.gov/pubmed/27647375
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2016.09.002
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