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ATP-competitive inhibitors block protein kinase recruitment to the Hsp90-Cdc37 system

Protein kinase clients are recruited to the Hsp90 molecular chaperone system via Cdc37, which simultaneously binds Hsp90 and kinases and regulates the Hsp90 chaperone cycle. Pharmacological inhibition of Hsp90 in vivo results in degradation of kinase clients, with a therapeutic effect in dependent t...

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Bibliografiske detaljer
Udgivet i:Nat Chem Biol
Main Authors: Polier, Sigrun, Samant, Rahul S., Clarke, Paul A., Workman, Paul, Prodromou, Chrisostomos, Pearl, Laurence H.
Format: Artigo
Sprog:Inglês
Udgivet: 2013
Fag:
Online adgang:https://ncbi.nlm.nih.gov/pmc/articles/PMC5695660/
https://ncbi.nlm.nih.gov/pubmed/23502424
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/nchembio.1212
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