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ACTR-45. A PHASE 1, MULTICENTER, OPEN-LABEL STUDY OF MARIZOMIB (MRZ) WITH TEMOZOLOMIDE (TMZ) AND RADIOTHERAPY (RT) IN NEWLY DIAGNOSED WHO GRADE IV MALIGNANT GLIOMA (GLIOBLASTOMA, ndGBM)

Proteasome inhibition sensitizes glioma cells to TMZ and RT, providing a novel therapeutic strategy for ndGBM. MRZ -- an irreversible, brain-penetrant, pan-proteasome inhibitor with anti-glioma preclinical activity -- is being evaluated in ndGBM patients (NCT02903069). The phase 1 study (MRZ at 0.55...

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Bibliografski detalji
Izdano u:Neuro Oncol
Glavni autori: Bota, Daniela, Mason, Warren, Kesari, Santosh, Piccioni, David, Aregawi, Dawit, Desjardins, Annick, Winograd, Benjamin, Reich, Steven D, Levin, Nancy, Trikha, Mohit
Format: Artigo
Jezik:Inglês
Izdano: Oxford University Press 2017
Teme:
Online pristup:https://ncbi.nlm.nih.gov/pmc/articles/PMC5692631/
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1093/neuonc/nox168.036
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