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Bifunctional aryliodonium salts for highly efficient radioiodination and astatination of antibodies

In this report we describe the development of an alternative approach to arylstannane chemistry for radiolabeling antibodies with radioiodine or astatine based on aryliodonium salts precursors. Bifunctional aryliodonium salts were designed and tested for the synthesis of (125)I and (211)At labeled p...

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Publicat a:Bioorg Med Chem
Autors principals: Guérard, F., Navarro, L., Lee, Y.-S., Roumesy, A., Alliot, C., Chérel, M., Brechbiel, M.W., Gestin, J.-F.
Format: Artigo
Idioma:Inglês
Publicat: 2017
Matèries:
Accés en línia:https://ncbi.nlm.nih.gov/pmc/articles/PMC5659727/
https://ncbi.nlm.nih.gov/pubmed/28964629
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1016/j.bmc.2017.09.022
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