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Activation of PKA in cell requires higher concentration of cAMP than in vitro: implications for compartmentalization of cAMP signalling

cAMP is a ubiquitous second messenger responsible for the cellular effects of multiple hormones and neurotransmitters via activation of its main effector, protein kinase A (PKA). Multiple studies have shown that the basal concentration of cAMP in several cell types is about 1 μM. This value is well...

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Pubblicato in:Sci Rep
Autori principali: Koschinski, Andreas, Zaccolo, Manuela
Natura: Artigo
Lingua:Inglês
Pubblicazione: Nature Publishing Group UK 2017
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Accesso online:https://ncbi.nlm.nih.gov/pmc/articles/PMC5658382/
https://ncbi.nlm.nih.gov/pubmed/29074866
https://ncbi.nlm.nih.govhttp://dx.doi.org/10.1038/s41598-017-13021-y
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